Miglitol

(British Approved Name, US Adopted Name, rINN)

Drug Nomenclature

International Nonproprietary Names (INNs) in main languages (French, Latin, Russian, and Spanish):

Synonyms: Bay-m-1099; Miglitol; Miglitoli; Miglitolum
USAN: Miglitol
INN: Miglitol [pINN (en)]
INN: Miglitol [pINN (es)]
INN: Miglitol [pINN (fr)]
INN: Miglitolum [pINN (la)]
INN: Миглитол [pINN (ru)]
Chemical name: (2R,3R,4R,5S)-1-(2-Hydroxyethyl)-2-(hydroxymethyl)piperidine-3,4,5-triol
Molecular formula: C8H17NO5 =207.2
CAS: 72432-03-2
ATC code: A10BF02

Adverse Effects and Precautions

As for alpha-glucosidase inhibitors in general (see Acarbose). Skin rash may occur. Miglitol should be used with caution in patients with renal impairment.

Interactions

As for alpha-glucosidase inhibitors in general (see Acarbose). Miglitol may reduce the bioavailability of propranolol and ranitidine.

Pharmacokinetics

Miglitol is completely absorbed at a dose of 25 mg, but only 50 to 70% is absorbed at a dose of 100 mg. It is not metabolised, and is excreted unchanged in the urine with a plasma elimination half-life of about 2 hours.

Uses and Administration

Miglitol is an alpha-glucosidase inhibitor similar in action to acarbose. It is given orally in the management of type 2 diabetes mellitus, alone or with a sulfonylurea. Usual initial doses are 25 mg three times daily with meals, increased if necessary to a maximum of 100 mg three times daily.

Proprietary Preparations

Austria: Diastabol

Czech Republic: Diastabol

France: Diastabol

Germany: Diastabol

Hungary: Diastabol

India: Diamig Mignar †

Mexico: Diastabol

Poland: Diastabol

Portugal: Diastabol Limarcan

Spain: Diastabol Plumarol

Sweden: Diastabol

Switzerland: Diastabol

USA: Glyset

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